DATASHEET
Formulation
White solid
Storage:
-20°C
Product Information:
A potent and selective GPR18 antagonist (IC50 = 0.279 M) exhibiting >36-fold selectivity against GPR55 and CB1 and 14-fold selectivity against CB2.1 Inhibits N-arachidonylglycine-induced acrosomal exocytosis in human spermatozoa indicating that GPR18 may be involved in physiological processes of human spermatozoa.2
Description:
CAS Number: 1627710-30-8<br></br>Chemical Name: (2Z)-2[[3-[(4-Chlorophenyl)methoxy]phenyl]methylene]-6,7-dihydro-5H-imidazo[2,1-b][1,3]thiazin-3(2H)-one<br></br>Molecular weight: 384.88<br></br>Formula: C20H17ClN2O2S<br></br>Solubility: DMSO (25 mg/ml)<br></br>Physical Properties: Pale-yellow solid<br></br>Purity: 98% by TLC NMR (Conforms)