DATASHEET
Formulation
Yellow solid
Storage:
-20°C
Product Information:
Tiagabine is a clinically useful anticonvulsant.1 It is also used to treat anxiety/panic disorder2 and neuropathic pain3. Tiagabine inhibits GABA-reuptake (IC50 [3H]GABA uptake = 67 nM) via inhibiting GABA transporter 1(GAT1) blocking both neuronal and glial GABA re-uptake.4,5
Description:
CAS Number: 145821-59-6<br></br>Chemical Name: (3R)-1-[4,4-Bis(3-methylthiophen-2-yl)but-3-enyl]piperidine-3-carboxylic acid hydrochloride<br></br>Molecular weight: 412.00<br></br>Formula: C20H25NO2S2·HCl<br></br>Solubility: DMSO (>25 mg/ml) Ethanol (>25 mg/ml) Water (>30 mg/ml)<br></br>Physical Properties: Off white or beige solid<br></br>Purity: >98% by HPLC NMR (Conforms)