bs-82821C
[Life Science]
S1RA
DATASHEET
Formulation White solid
Storage: -20°C
Product Information:
S1RA (E-52862) is a potent and selective 1 antagonist with weak binding at 2 (IC50’s: 1 = 17nM, 2 = 9300nM).1,2 S1RA abolished mechanical and thermal hyperalgesia in mice with carrageenan-induced acute inflammation by enhancing the action of endogenous opioid peptides of immune origin in a 1 dependent manner.3 BD1063 potentiated µ-opioid antinociception in mice in a -dependent manner.4 S1RA displayed neuroprotective effects in a mouse model of ischemic stroke.5
Description:
CAS Number: 1265917-14-3<br></br>Chemical Name: 4-{2-[5-Methyl-1-(napthalen-2-yl)-1H-pyrazol-3-yloxy]ethyl}morpholine hydrochloride<br></br>Molecular weight: 373.88<br></br>Formula: C20H23N3O2·HCl<br></br>Solubility: DMSO (>25 mg/ml)<br></br>Physical Properties: Off-white solid<br></br>Purity: 98% by HPLC NMR (Conforms)
Size: 5 mg, 25 mg5 mg, 25 mg
Applications: Life Science()
For research use only. Not intended for diagnostic or therapeutic use.