bs-82758C [Life Science]
GSK6853
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Formulation Off-white solid

Storage: -20°C

Product Information:

Very potent (pIC50 = 8.6 vs full length protein, 7.7 in cellular assays) inhibitor of Bromodomain and PHD Finger-containing 1 (BRPF1). It displayed >1600-fold selectivity over other bromodomains.

Description:

CAS Number: 1910124-24-1<br></br>Chemical Name: N-[1,3-Dimethyl-6-[(2R)-2-methylpiperazin-1-yl]-2-oxobenzimidazol-5-yl]-2-methoxybenzamide<br></br>Molecular weight: 409.49<br></br>Formula: C22H27N5O3<br></br>Solubility: DMSO (25 mg/ml); ethanol (25 mg/ml)<br></br>Physical Properties: White solid<br></br>Purity: 98% by HPLC NMR (Conforms)

Size: 5 mg, 25 mg5 mg, 25 mg

Applications: Life Science()

For research use only. Not intended for diagnostic or therapeutic use.