bs-82694C
[Life Science]
DJ-V 159
DATASHEET
Formulation White solid
Storage: RT
Product Information:
GPRC6A is the receptor for osteocalcin as well as structurally unrelated ligands including L-amino acids, cations and anabolic steroids.1 GPRC6A is a potential therapeutic target for treating type 2 diabetes.2 DJ-V 159 is an agonist at GPRC6A which activates ERK and upregulates cAMP levels in HEK-193 cells expressing GPRC6A It stimulates insulin secretion in mouse -cells and lowers blood glucose in mouse models.3
Description:
CAS Number: 2253744-53-3<br></br>Chemical Name: N1,N3-Bis(4-cyano-3-(trifluoromethyl)phenyl)isophthalamide<br></br>Molecular weight: 502.37<br></br>Formula: C24H12F6N4O2 <br></br>Solubility: DMSO (60 mg/ml)<br></br>Physical Properties: Off-white solid<br></br>Purity: 98% by TLC NMR (Conforms)
Size: 5 mg, 25 mg5 mg, 25 mg
Applications: Life Science()
For research use only. Not intended for diagnostic or therapeutic use.