DATASHEET
Formulation
White solid
Storage:
-20°C
Product Information:
Varenicline is a partial agonist of the α4β2 neuronal nicotinic acetylcholine receptor (EC50 = 2.3 µM) and a full agonist at α7 neuronal nicotinic receptors.1 Clinically useful smoking cessation agent.2,3
Description:
CAS Number: 375815-87-5<br></br>Chemical Name: 7,8,9,10-Tetrahydro-6H-6,10-methanoazepino[4,5-g]quinoxaline tartrate:7,8,9,10-Tetrahydro-6,10-methano-6H-pyrazino(2,3-h)(3)benzazepine tartrate<br></br>Molecular weight: 361.35<br></br>Formula: C13H13N3·C4H6O6<br></br>Solubility: DMSO (18 mg/ml) Water (35 mg/ml)<br></br>Physical Properties: Yellow solid<br></br>Purity: 99% by HPLC, NMR (Conforms)