DATASHEET
Formulation
Off-white solid
Storage:
RT
Product Information:
A semi-synthetic ergoline derivative which acts as a partial dopamine D2 agonist and 5HT2B/2C receptor antagonist. Displays antiparkinsonian effects in MPTP-treated cynomolgus monkeys1. Partial agonist at recruitment of -arrestin2 to the D2 receptor2. Ameliorates monocrotaline-induced pulmonary hypertension in rats3.
Description:
CAS Number: 37686-84-3<br></br>Chemical Name: S(+)-N,N-Diethyl-N′([8α]-6-methylergolin-8-yl)urea<br></br>Molecular weight: 340.47<br></br>Formula: C20H28N4O<br></br>Solubility: DMSO or Ethanol<br></br>Physical Properties: White solid<br></br>Purity: 98% by TLC, NMR (conforms)