DATASHEET
Formulation
White or off-white solid
Storage:
-20°C
Product Information:
Selective protein kinase G inhibitor (Ki =0.23, 4 and >10 μM for PKG, PKC and PKA respectively1. Arrests human skin fibroblast cell cycle after the G0/G1 boundary2. Abolishes the cGMP-induced relaxation in smooth muscle cells (IC50=60 nM)3. Cell permeable.
Description:
CAS Number: 126643-37-6<br></br>Chemical Name: <br></br>Molecular weight: 495.53<br></br>Formula: C29H25N3O5<br></br>Solubility: DMSO (25 mg/ml) DMF (20 mg/ml)<br></br>Physical Properties: White or off white solid<br></br>Purity: 98% by TLC, NMR (Conforms)