bs-82285C [Life Science]
TC-E 5003
www.biossusa.com
[email protected]
800.501.7654 [DOMESTIC]
+1.781.569.5821 [INTERNATIONAL]
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Formulation Off-white solid

Storage: -20°C

Product Information:

Selective protein arginine methyltransferase 1 (PRMT1) inhibitor, IC50 = 1.5 μM. Displays no activity against CARM1 and Set7/9 methyltransferases. Inhibits growth of MCF7a breast cancer cells and LNCaP prostate cancer cells. Blocks androgen-induced gene expression in LNCaP cells1.

Description:

CAS Number: 17328-16-4<br></br>Chemical Name: N,N’-(Sulfonyldi-4,1-phenylene)bis(2-chloroacetamide)<br></br>Molecular weight: 401.26<br></br>Formula: C16H14Cl2N2O4S<br></br>Solubility: DMSO 50 mg/ml<br></br>Physical Properties: Brown solid<br></br>Purity: 98% by HPLC NMR (Conforms)

Size: 50 mg, 250 mg50 mg, 250 mg

Applications: Life Science()

For research use only. Not intended for diagnostic or therapeutic use.