DATASHEET
Formulation
Light brown solid
Storage:
-20°C
Product Information:
RVX-208 is a potent BET bromodomain antagonist with IC50 of 0.510 μM for BD2, with approximately 170-fold selectivity over BD11,2. Increases apolipoprotein A-1 and HDL cholesterol in vitro and in vivo3. Reduces atherosclerosis4.
Description:
CAS Number: 1044870-39-4<br></br>Chemical Name: 2-[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]-5,7-dimethoxy-4(3H)-quinzolinone<br></br>Molecular weight: 370.41<br></br>Formula: C20H22N2O5<br></br>Solubility: DMSO (75 mg/ml) Ethanol (4 mg/ml)<br></br>Physical Properties: White solid<br></br>Purity: 98% by TLC, NMR (Conforms)