DATASHEET
Formulation
Beige solid
Storage:
RT
Product Information:
Potent and selective ATP-competitive inhibitor of protein kinase D (PKD). IC50=3.2, 0.6 and 0.7 μM for PKD1, 2 and 3 respectively. Inhibits phorbol ester-induced PKD activation in LNCaP prostate cancer cells. Cell permeable.
Description:
CAS Number: 638156-11-3<br></br>Chemical Name: 5-(3-Chlorophenyl)-N-[4-(4-morpholinylmethyl)phenyl]-2-furancarboxamide<br></br>Molecular weight: 396.88<br></br>Formula: C22H21ClN2O3<br></br>Solubility: DMSO (50 mg/ml) Ethanol (8 mg/ml)<br></br>Physical Properties: Tan solid<br></br>Purity: 98% by TLC, NMR (Conforms)