DATASHEET
Formulation
White solid
Storage:
RT
Product Information:
Prostaglandin E2 (EP1 receptor) antagonist (pA2=6.5, guinea pig ileum muscle strip assay )1,4. Possesses analgesic activity in vivo (rodent ED50= 6.8 mg/kg)1,2,4. Does not inhibit COX11 and does not block PGE1 induced hyperalgesia3.
Description:
CAS Number: 146033-02-5<br></br>Chemical Name: 8-Cholrodibenz(Z)[b,f]oxazepine-10(11H)-carboxylic acid 2-[1-oxo-3-(4-pyridinyl)propyl]hydrazide hydrochloride<br></br>Molecular weight: 459.34<br></br>Formula: C22H19ClN4O3 ยท HCl<br></br>Solubility: DMSO (25 mg/ml) Water (25 mg/ml)<br></br>Physical Properties: White solid<br></br>Purity: 98% by TLC, NMR (Conforms)