bs-82058C
[Life Science]
BCTC
DATASHEET
Formulation Off-white solid
Storage: RT
Product Information:
Vanilloid receptor I (TRPV1) antagonist, IC50 = 35 nM for capsaicin-induced and 6 nM for acid-induced TRPV1 activation. Displays analgesic activity in rat models of neuropathic pain. Orally active and cell permeable.
Description:
CAS Number: 393514-24-4<br></br>Chemical Name: 4-(3-Chloro-2-pyridinyl)-N-[4-(1,1-dimethylethyl)phenyl]-1-piperazinecarboxamide<br></br>Molecular weight: 372.9<br></br>Formula: C20H25ClN4O<br></br>Solubility: DMSO (25 mg/ml) Ethanol (15 mg/ml)<br></br>Physical Properties: Off-white solid<br></br>Purity: 98% by TLC [ 2% CH3OH in CH2Cl2; Rf = 0.25] NMR Conforms
Size: 10 mg, 50 mg10 mg, 50 mg
Applications: Life Science()
For research use only. Not intended for diagnostic or therapeutic use.