DATASHEET
Formulation
yellow solid (MP = 209-211°C)
Storage:
RT
Product Information:
Reversible, competitive inhibitor of IKK2 (IC50 = 11.2 µM). Has not been demonstrated to inhibit other IKK isoforms, or other kinases. Displays dose-dependent inhibition of the transcription of NK-κB dependent genes in cell culture1.
Description:
CAS Number: 354812-17-2<br></br>Chemical Name: 5-(Thien-3-yl)-3-aminothiophene-2-carboxamide<br></br>Molecular weight: 224.3<br></br>Formula: C9H8N2OS2<br></br>Solubility: DMSO (25 mg/ml)<br></br>Physical Properties: yellow solid (MP = 209-211°C)<br></br>Purity: 98% by TLC [5% methanol in methylene chloride; Rf= 0.27] NMR conforms