bs-80291C
[Life Science]
RVX-208
DATASHEET
Formulation powder
Storage: -20°C
Product Information:
Molecular Weight:370.41
Formula:C20H22N2O5
Purity:>98%
Solubility:Soluble in DMSO (up to 75 mg/ml) or in Ethanol (up to 4 mg/ml).
Chemical Name:2-[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]-5,7-dimethoxy-4(3H)-quinzolinone
Formula:C20H22N2O5
Purity:>98%
Solubility:Soluble in DMSO (up to 75 mg/ml) or in Ethanol (up to 4 mg/ml).
Chemical Name:2-[4-(2-hydroxyethoxy)-3,5-dimethylphenyl]-5,7-dimethoxy-4(3H)-quinzolinone
Description:
RVX-208 is a potent BET bromodomain antagonist with IC50 of 0.510 μM for BD2, with approximately 170-fold selectivity over BD11,2. Increases apolipoprotein A-1 and HDL cholesterol in vitro and in vivo3. Reduces atherosclerosis4.
Size: 5 mg, 25 mg5 mg, 25 mg
Applications: Life Science()
For research use only. Not intended for diagnostic or therapeutic use.