DATASHEET
Formulation
powder
Storage:
RT
Product Information:
Molecular Weight:537.1
Formula:C26H26ClN2O3S2 ยท Na
Purity:>98%
Solubility:Soluble in DMSO (up to 50 mg/ml).
Chemical Name:5-(3-(2-(7-Chloroquinolin-2-yl)ethenyl)phenyl)-8-dimethylcarbamyl-4,6-dithiaoctanoic acid, sodium salt
Description:
Potent (EC50 = 1.3nM) and selective Leukotriene D4 antagonist(LTD4)1 displaying inverse agonist activity2, Blocks binding of LTD4 to human (Ki = 0.22 nM) and guinea pig (Ki = 2.1 nM) lung membranes. Selective for the CysLT1 receptor. Multidrug resistance protein 1 (MRP1) inhibitor.3